The clinically-tested S1P receptor agonists, FTY720 and BAF312, demonstrate subtype-specific bradycardia (S1P₁) and hypertension (S1P₃) in rat. Fryer RM, Muthukumarana A, Harrison PC, Nodop Mazurek S, Chen R R, Harrington KE, Dinallo RM, Horan JC, Patnaude L, Modis LK, et al. PLoS One. 2012; 7(12):e52985. Epub 2012 Dec 28. PMID: 23285242. Abstract CommentRecommendBookmarkWatch