Structure-Kinetics Relationships - an overlooked parameter in hit-to-lead optimization: a case of cyclopentylamines as CCR2 antagonists. Vilums M, Zweemer A, Yu Z, de Vries H, Hillger J, Wapenaar H, Bollen I, Barmare F, Gross RS, Clemens JJ, et al. J Med Chem. 2013 Sep 12. PMID: 24028535. Abstract CommentRecommendBookmarkWatch