When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists.
Vilums M, Zweemer AJM, Barmare F, van der Gracht AMF, Bleeker DCT, Yu Z, de Vries H, Gross R, Clemens J, Krenitsky P, et al.
Eur J Med Chem. 2015 Feb 2; 93C:121-134. PMID: 25666912.Abstract